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Characterization of Stable Pyrazole Derivatives of Curcumin with Improved Cytotoxicity on Osteosarcoma Cell Lines
Feriotto, G.; Rondanin, R.; Marchetti, P.; Tagliati, F.; Beninati, S.; Tabolacci, C.; Grusi, E.; Aguzzi, S.; Mischiati, C.     details >>
LIFE
Vol. 13, No. 2, pp: 431-1-431-14, Anno: 2023

Cytotoxicity of Isoxazole Curcumin Analogs on Chronic Myeloid Leukemia-Derived K562 Cell Lines Sensitive and Resistant to Imatinib
Feriotto, G.; Marchetti, P.; Rondanin, R.; Tagliati, F.; Aguzzi, S.; Beninati, S.; Casciano, F.; Tabolacci, C.; Mischiati, C.     details >>
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES
Vol. 24, No. 3, pp: 1-17, Anno: 2023

Pro‑apoptotic activity of novel synthetic isoxazole derivatives exhibiting inhibitory activity against tumor cell growth in vitro
Lampronti, I.; Simoni, D.; Rondanin, R.; Baruchello, R.; Scapoli, C.; Finotti, A.; Borgatti, M.; Tupini, C.; Gambari, R.     details >>
ONCOLOGY LETTERS
Vol. 20, No. 5, pp: 151-1-151-11, Anno: 2020

New TRAP1 and Hsp90 chaperone inhibitors with cationic components: Preliminary studies on mitochondrial targeting
Rondanin, R; Lettini, G; Oliva, P; Baruchello, R; Costantini, C; Trapella, C; Simoni, D; Bernardi, T; Sisinni, L; Pietrafesa, M; Ponterini, G; Costi, M P; Vignudelli, T; Luciani, R; Matassa, D S; Esposito, F; Landriscina, M     details >>
BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS
Vol. 28, No. 13, pp: 2289-2293, Anno: 2018

Design, synthesis, in vitro antiproliferative activity and apoptosis-inducing studies of 1-(3',4',5'-trimethoxyphenyl)-3-(2'-alkoxycarbonylindolyl)-2-propen-1-one derivatives obtained by a molecular hybridisation approach
Preti, Delia; Romagnoli, Romeo; Rondanin, Riccardo; Cacciari, Barbara; Hamel, Ernest; Balzarini, Jan; Liekens, Sandra; Schols, Dominique; Estévez-Sarmiento, Francisco; Quintana, José; Estévez, Francisco     details >>
JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Vol. 33, No. 1, pp: 1225-1238, Anno: 2018

Effects of Pimozide Derivatives on pSTAT5 in K562 Cells
Rondanin, Riccardo; Simoni, Daniele; Maccesi, Martina; Romagnoli, Romeo; Grimaudo, Stefania; Pipitone, Rosaria Maria; Meli, Maria; Cascio, Antonio; Tolomeo, Manlio     details >>
CHEMMEDCHEM
Vol. 12, No. 15, pp: 1183-1190, Anno: 2017

Arylamidonaphtalene sulfonate compounds as a novel class of heparanase inhibitors
Rondanin, Riccardo; Fochi, Sara; Baruchello, Riccardo; Bernardi, Tatiana; Oliva, Paola; Semeraro, Floriana; Simoni, Daniele; Giannini, Giuseppe     details >>
BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS
Vol. 27, No. 18, pp: 4421-4425, Anno: 2017

Novel iodoacetamido benzoheterocyclic derivatives with potent antileukemic activity are inhibitors of STAT5 phosphorylation
Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Lopez Cara, Carlota; Rondanin, Riccardo; Simoni, Daniele; Hamel, Ernest; Grimaudo, Stefania; Pipitone, Rosaria Maria; Meli, Maria; Tolomeo, Manlio     details >>
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Vol. 108, No. 1, pp: 39-52, Anno: 2016

Hemiasterlin derivative (R)(S)(S)-BF65 and Akt inhibitor MK-2206 synergistically inhibit SKOV3 ovarian cancer cell growth
Lai, Wei Ting; Cheng, Kai Lin; Baruchello, Riccardo; Rondanin, Riccardo; Marchetti, Paolo; Simoni, Daniele; Lee, Ray M.; Guh, Jih Hwa; Hsu, Lih Ching     details >>
BIOCHEMICAL PHARMACOLOGY
Vol. 113, No. 1, pp: 12-23, Anno: 2016

A novel hybrid drug between two potent anti-tubulin agents as a potential prolonged anticancer approach
Marchetti, Paolo; Pavan, Barbara; Simoni, Daniele; Baruchello, Riccardo; Rondanin, Riccardo; Mischiati, Carlo; Feriotto, Giordana; Ferraro, Luca Nicola; Hsu, Lih Ching; Lee, Ray M.; Dalpiaz, Alessandro     details >>
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES
Vol. 91, No. 1, pp: 50-63, Anno: 2016

Inhibition of activated STAT5 in Bcr/Abl expressing leukemia cells with new pimozide derivatives.
Rondanin, Riccardo; Simoni, Daniele; Romagnoli, Romeo; Baruchello, Riccardo; Marchetti, Paolo; Costantini, Cristiana; Fochi, Sara; Padroni, Giacomo; S., Grimaudo; R. M., Pipitone; M., Meli; M., Tolomeo     details >>
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Vol. 24, No. 1, pp: 4568-4574, Anno: 2014

4,5,6,7-Tetrahydro-isoxazolo-[4,5-c]-pyridines as a new class of cytotoxic Hsp90 inhibitors
Baruchello, Riccardo; Simoni, Daniele; Marchetti, Paolo; Rondanin, Riccardo; Mangiola, Stefania; Costantini, Cristiana; M., Meli; G., Giannini; L., Vesci; V., Carollo; T., Brunetti; G., Battistuzzi; M., Tolomeo; W., Cabri     details >>
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Vol. 76, No. 1, pp: 53-60, Anno: 2014

Development of hemiasterlin derivatives as potential anticancer agents that inhibit tubulin polymerization and synergize with a stilbene tubulin inhibitor.
L., Hsu; D. E., Durrant; C., Huang; N., Chi; Baruchello, Riccardo; Rondanin, Riccardo; Rullo, Cinzia; Marchetti, Paolo; Grisolia, Giuseppina; Simoni, Daniele; R. M., Lee     details >>
INVESTIGATIONAL NEW DRUGS
Vol. 30, No. 1, pp: 1379-1388, Anno: 2012

Novel 3,4-isoxazolediamides as potent inhibitors of chaperone heat shock protein 90.
Baruchello, Riccardo; Simoni, Daniele; Grisolia, Giuseppina; G., Barbato; Marchetti, Paolo; Rondanin, Riccardo; Mangiola, Stefania; G., Giannini; T., Brunetti; D., Alloatti; G., Gallo; A., Ciacci; L., Vesci; M., Castorina; F. M., Milazzo; M. L., Cervoni; M. B., Guglielmi; M., Barbarino; R., Foderà; C., Pisano; W., Cabri     details >>
JOURNAL OF MEDICINAL CHEMISTRY
Vol. 54, No. 1, pp: 8592-8604, Anno: 2011

Synthesis and biological activity of a novel class nicotinic acetylcholine receptors (nAChRs) ligands structurally related to anatoxin-a.
Simoni, Daniele; Rondanin, Riccardo; Marchetti, Paolo; Rullo, Cinzia; Baruchello, Riccardo; Grisolia, Giuseppina; G., Barbato; R., Giovannini; C., Marchioro; A. M., Capelli; C., Virginio; A., Bozzoli; Borea, Pier Andrea; Merighi, Stefania; D., Donati     details >>
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Vol. 21, No. 1, pp: 5423-5427, Anno: 2011

Versatile Synthesis of New Cytotoxic Agents Structurally Related to Emiasterlins
Simoni, Daniele; R. M., Lee; D. E., Durrant; N., Chi; Baruchello, Riccardo; Rondanin, Riccardo; Rullo, Cinzia; Marchetti, Paolo     details >>
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Vol. 20, No. 1, pp: 3431-3435, Anno: 2010

Inhibition of cell proliferation by a resveratrol analog in human pancreatic and breast cancer cells
Y. B., Hong; H. J., Kang; H. J., Kim; E. M., Rosen; S., Dakshanamurthy; Rondanin, Riccardo; Baruchello, Riccardo; Grisolia, Giuseppina; Simoni, Daniele; I. B. a., E.     details >>
EXPERIMENTAL AND MOLECULAR MEDICINE
Vol. 41, No. 3, pp: 151-160, Anno: 2009

Design, synthesis and biological evaluation of novel stilbene-based antitumor agents
Simoni, Daniele; Francesco Paolo, Invidiata; Eleopra, Marco; Marchetti, Paolo; Rondanin, Riccardo; Baruchello, Riccardo; Grisolia, Giuseppina; Ashutosh, Tripathi; Glen E., Kellogg; David, Durrant; Ray M., Lee     details >>
BIOORGANIC & MEDICINAL CHEMISTRY
Vol. 17, No. 2, pp: 512-522, Anno: 2009

Novel terphenyls and 3,5-diaryl isoxazole derivatives endowed with growth supporting and antiapoptotic properties
Simoni, Daniele; Rondanin, Riccardo; Baruchello, Riccardo; Rizzi, Michele; Grisolia, Giuseppina; Eleopra, Marco; Stefania, Grimaudo; Antonietta Di, Cristina; Maria Rosaria, Pipitone; Maria Rita, Bongiorno; Mario, Aricò; Francesco Paolo, Invidiata; Manlio, Tolomeo     details >>
JOURNAL OF MEDICINAL CHEMISTRY
Vol. 51, No. 15, pp: 4796-4803, Anno: 2008

Design, synthesis, and biological evaluation of novel aminobisphosphonates possessing an in vivo antitumor activity through a γδ-T lymphocytes-mediated activation mechanism
Simoni, Daniele; Nicola, Gebbia; Francesco Paolo, Invidiata; Eleopra, Marco; Marchetti, Paolo; Rondanin, Riccardo; Baruchello, Riccardo; Stefano, Provera; Carla, Marchioro; Manlio, Tolomeo; Luciana, Marinelli; Vittorio, Limongelli; Ettore, Novellino; Aaron, Kwaasi; James, Dunford; Simona, Buccheri; Nadia, Caccamo; Francesco, Dieli     details >>
JOURNAL OF MEDICINAL CHEMISTRY
Vol. 51, No. 21, pp: 6800-6807, Anno: 2008

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